2024
Masahiro Abe,* Mai Takano, Akiho Mizukami, Tetsutaro Kimachi, Kiyofumi Inamoto*
The Journal of Organic Chemistry, accepted for publication, 2024
Masahiro Abe,* Megumu Kawamoto, Akiho Mizukami, Tetsutaro Kimachi, Kiyofumi Inamoto*
The Journal of Organic Chemistry, 89(14), 10037-10046, 2024
Masahiro Abe,* Akiho Mizukami, Emi Yoshida, Tetsutaro Kimachi, Kiyofumi Inamoto*
RSC Advances, 14(2), 808-811, 2024
2023
Masahiro Abe,* Honoka Jitsumatsu, Mikoto Araki, Akiho Mizukami, Tetsutaro Kimachi, Kiyofumi Inamoto*
Synthesis, 55(19), 3121-3128, 2023
2022
Masahiro Abe,* Megumu Kawamoto, Mayu Inoue, Tetsutaro Kimachi, Kiyofumi Inamoto*
Organic Letters, 24(31), 5684-5687, 2022
Masahiro Abe,* Yuka Yokoi, Aoi Hirata, Yumeno Matsuoka, Tetsutaro Kimachi, Kiyofumi Inamoto*
Chemical Communications, 58(53), 7416-7418, 2022
Masahiro Abe,* Sayasa Nitta, Erina Miura, Tetsutaro Kimachi, Kiyofumi Inamoto*
The Journal of Organic Chemistry, 87(6), 4460-4467, 2022
2021
Masahiro Abe,* Kaho Ueta, Saki Tanaka, Tetsutaro Kimachi, Kiyofumi Inamoto*
RSC Advances, 11(43), 26988-26991, 2021
2020
Noboru Hayama, Yusuke Kobayashi, Eriko Sekimoto, Anna Miyazaki, Kiyofumi Inamoto, Tetsutaro Kimachi, Yoshiji Takemoto*
Chemical Science, 11(21), 5572-5576, 2020
2019
Evaluation of molecularly imprinted polymers for chlorpromazine and bromopromazine
prepared by multi-step swelling and polymerization method -The application for the determination of chlorpromazine and its metabolites in rat plasma by column-switching LC
Kanae Nishimura, Noboru Okamuira, Tetsutaro Kimachi, Jun Haginaka* Journal of Pharmaceutical and Biomedical Analysis, 174, 248-255, 2019 |
Retention and molecular-recognition mechanisms of molecularly imprinted
polymers for promazine derivatives
Jun Haginaka*, Kanae Nishimura, Tetsutaro Kimachi, Kiyofumi Inamoto, Yoshiji Takemoto, Yusuke Kobayashi Talanta, 205, 120149, 2019 |
Rhodium-catalyzed Synthesis of Benzo[b]thiophene-3-carboxamides via Cyclization
of (ortho-Alkynyl)phenyl Sulfides in the Presence of Isocyanates
Akiho Mizugami, Maika Tsugita, Mako Shimora, Saki Tanaka, Noboru Hayama, Tetsutaro Kimachi, Kiyofumi Inamoto* Chemistry Letters, 48(5), 12014, 2019 |
Catalytic asymmetric aza-Michael addition of fumaric monoacids with multifunctional
thiourea / boronic acids
Kenichi Michigami, Hiroki Murakami, Takeru Nakamura, Noboru Hayama, Yoshiji Takemoto* Organic&Biomolecular Chemistry, 17(9), 2331-2335, 2019 |
Inhibition of angiogenesis and tumor growth by a novel 1,4-naphthoquinone
derivative
Hiroko Murata, Tomohiro Shinya, Mariko Sakanaka, Satoru Takahashi, Arisa Nishiuchi, Tokutaro Ogata, Noboru Hayama, Tetsutaro Kimachi, Kenichi Toda, Satoru Takahashi Drug Development Research, 80(3), 395-402, 2019 |
2018
Construction of cyclic ether-fused tricyclic naphtoquinone derivatives
by intramolecular cyclization reaction
Tokutaro Ogata, Tetsutaro Kimachi Heterocycles, 97, 107-140, 2018 |
Mechanistic Insight into Asymmetric Hetero-Michael Addition of α,β-Unsaturated
Carboxylic Acids Catalyzed by Multifunctional Thioureas
Noboru Hayama, Ryuta Kuramoto, Kazuya Nishibayashi, Yusuke Kobayashi, Yoshiji Takemoto*, Tamas Foldes, Imre Papai* Journal of the American Chemical Society, 140 (38), 12216–12225, 2018 |
PET probe detecting non-small cell lung cancer susceptible to epidermal
growth factor receptor tyrosine kinase inhibitor therapy
Akira Makino, Anna Miyazaki, Ayaka Tomoike, Masahiro Ono, Hiroyuki Kimura, Kenji Arimitsu, Masahiro Hirata, Yoshiro Ohmoto, Ryuichi Nishii et al. Bioorganic&Medicinal Chemistry, 26 (8), 1609–1613 (2018) |
2017
Copper-catalyzed intramolecular C-H amination: a new entry to substituted
xanthine derivatives
Maki Shimizu, Noboru Hayama, Tetsutaro Kimachi, Kiyofumi Inamoto* Synthesis, 49 (18), 4183-4190, 2017 |
Simultaneous functionalization and cyclization of 2-ethynylaniline derivatives
to indoles
Hiroya Kou, Shin Itoh, Kiyofumi Inamoto, Hiroki Shigehisa, Takao Sakamoto Heterocycles, 95, 920-933, 2017 |
(18)F-Labeled Pyrido[3,4-d]pyrimidiine as an Effective Prode for Imaging
of L858R Mutant Epidermal Growth Factor Receptor
Hiroyuki Kimura, Haruka Okuda, Masumi Ishiguro, Kenji Arimitsu, Akira Makino, Ryuichi Nishii, Anna Miyazaki, Yusuke Yagi, Hiroyuki Watanabe et al. ACS Medicinal Chemistry Letters, 8 (4), 418–422, 2017 |
2016
Unusual, chemoselective etherification of 2-hydroxy-1,4-naphthoquinone
derivatives utilizing alkoxymethyl chlorides: scope, mechanism and application
to the synthesis of biologically active natural product (±)-lantalucratin
C
Tokutaro Ogata, Tomoyo Yoshida, Maki Shimizu, Manami Tanaka, Chie Fukuhara, Junko Ishii,
Arisa Nishiuchi, Kiyofumi Inamoto, Tetsutaro Kimachi Tetrahedron, 72 (11), 1423–1432, 2016
|
Rhodium-Catalyzed Cyclization of 2-Ethynylanilines in the Presence of Isocyanates:
Approach toward Indole-3-carboxamides Akiho Mizukami, Yumi Ise, Tetsutaro Kimachi, Kiyofumi Inamoto* Organic
Letters, 18 (4), 748–751, 2016
|
Development of hemiacetal esterified levofloxacin to prevent chelation
with metal-containing drugs
Toru Otori, Sumio Matzno, Atushi Kawase, Masahiro Iwaki, Tetsutaro Kimachi, Kenji Nishiwaki, William C. Figoni, Ryuta Tominaga, Mai Asahide, Mayumi Nishikata, Yoshikazu Ishii, Kenji Mathuyama* Journal of Pharmacy and Pharmacology, 68 , 1527–1534, 2016 |
Chiral Intergrated Catalysts Composed of Bifunctional Thiourea and Arylboronic
Acid: Asymmetric Aza-Michael Addition of α, β-Unsaturated Carboxylic Acids
Noboru Hayama, Takumi Azuma, Yusuke Kobayashi, Yoshiji Takemoto* Chemical&Pharmaceutical Bulletin, 64(7) , 704-17, 2016 |
Palladiium-Catalyzed Highly Chemoselective Intramolecular C-H Aminocarbonylation
of Phenethylamines to Six-Membered Benzolactams
Hiroshi Taneda, Yoshinori Kondo*, Kiyofumi Inamoto* Organic Letters, 18(11) , 70-17, 2016 |
2015
Unusual O-Alkylation of 2-Hydroxy-1,4-naphthoquinone Utilizing Alkoxymethyl
Chlorides Tokutaro Ogata, Tomoyo Yoshida, Manami Tanaka, Chie Fukuhara, Maki Shimizu, Junko Ishii,
Arisa Nishiuchi, Kiyofumi Inamoto, Tetsutaro Kimachi Chemical & Pharmaceutical Bulletin, 63, 485–488, 2015
|
The first enantioselective total synthesis of lantalucratin C and determination
of its absolute configuration Tokutaro Ogata, Manami Tanaka, Momoe Ishigaki, Maki Shimizu, Arisa Nishiuchi, Kiyofumi Inamoto, Tetsutaro Kimachi Tetrahedron, 71 (38), 6672–6680, 2015
|
Highly Enantioselective (−)-Sparteine-Mediated Lateral Metalation-Functionalization
of Remote Silyl Protected ortho-Ethyl N,N-Dialkyl Aryl O-Carbamates
Jurg Fassler, J. Adam McCubbin, Anna Roglans, Tetsutaro Kimachi, Joshua W. Hollett, Roland W. Kunz, Michael Tinkl, Yousheng Zhang, Ruiyao Wang, Michae Campbell, Victor Snieckus The Journal of Organic Chemistry, 80 (7), 3368–3386 (2015) > |
2014
A diversity-oriented synthesis of caroverine derivatives via TEMPO-promoted
aerobic oxidative C–N bond formation
Yusuke Kobayashi, Yusuke Suzuki, Tokutaro Ogata, Tetsutaro Kimachi, Yoshiji Takemoto* Tetrahedron Letters, 55 (22), 3299–3301, 2014
|
Studies on the oxidative cyclization of 3-hydroxy-1,2,4-trialkoxynaphthalenes and synthetic application for the biologically active natural compound:
rhinacanthone
Tokutaro Ogata, Misae Doe, Aya Matsubara, Eri Torii, Chiaki Nishiura, Arisa Nishiuchi, Yusuke Kobayashi, Tetsutaro Kimachi* Tetrahedron, 70 (2), 502–509, 2014
|
2013
Total synthesis of (±)-lantalucratins A and B by CAN-mediated oxidative
cyclization
Tokutaro Ogata, Yoshiko Sugiyama, Saki Ito, Kazuha Nakano, Eri, Torii, Arisa Nishiuch, Tetsutaro Kimachi* Tetrahedron, 69, 10470–10476, 2013
|
2012
Catalytic Asymmetric Synthesis of (S)-Laudanosine by Hydroamination
Tokutaro Ogata, Tetsutaro Kimachi, Ken-ichi Yamada, Yasutomo Yamamoto, Kiyoshi Tomioka* Heterocycles, 86, 469–485, 2012
|
Organocatalyzed Isomerization of α-Substituted Alkynoates into Trisubstituted
Allenoates by Dynamic Kinetic Resolution
Tsubasa Inokuma, Masaya Furukawa, Yusuke Suzuki, Tetsutaro Kimachi, Yusuke Kobayashi, Yoshiji Takemoto* ChemCatChem, 4 (7), 983–985, 2012
|
2011
Highly efficient synthesis of quinoxalinone-N-oxide via tandem nitrosation/aerobic oxidative C–N bond formation
Yusuke Kobayashi,* Mami Kuroda, Natsuki Toba, Mari Okada, Rie Tanaka, Tetsutaro Kimachi* Organic Letters,13,6280–6283, 2011
|
Asymmetric total synthesis of biologically active (–)-dehydroiso-β-lapachone and the determination of its absolute configuration Tetsutaro
Kimachi,* Eri Torii, Yusuke Kobayashi, Misae Doe, Motoharu Ju-ichi Chemical & Pharmaceutical Bulletin, 59, 753–756, 2011
|
An efficient construction of nitrogen-containing
heterocycles utilizing CN functional groups and its application to the synthesis
of natural products Yusuke
Kobayashi*
Yakugaku Zasshi, 131, 1037–1046, 2011 |
α-Dimethylaminomethylenation-induced Houben–Hoesch-type cyclization of cyanoacetanilides:
A practical synthesis of 3-formyl-4-hydroxyquinolin-2(1H)-ones Yusuke Kobayashi,* Terue Nakatani, Rie Tanaka, Mari Okada, Eri Torii, Takashi Harayama, Tetsutaro Kimachi* Tetrahedron, 67, 3457–3463, 2011 |
Regioselective ring-opening
reaction of unsymmetrical 2,3-diaryl epoxides via catalytic hydrogenolysis with
Pd(0)EnCatTM Tetsutaro
Kimachi,*
Hiroyo Nagata, Yusuke Kobayashi, Kaori Takahashi, Eri Torii, Motoharu Ju-ichi Synlett, (3), 365–368 (2011) |
Synthetic studies of
salinosporamide A through the intramolecular hydroamidation of alkynes Haruhi
Kamisaki, Yusuke Kobayashi, Tetsutaro Kimachi, Yoshizumi Yasui,
Yoshiji Takemoto* Journal of Organometallic
Chemistry,
696, 42–45 (2011) |
Asymmetric Darzens-type epoxidation
via chiral ammonium ylides Hiroyo
Kinoshita, Akiko Ihoriya, Motoharu Ju-ichi, Tetsutaro Kimachi* Synlett, (15), 2330–2334
(2010) |
Enantioselective reduction of ketones
and imines catalyzed by (CN-Box)ReV–oxo complexes Kristine A.
Nolin, Richard W. Ahn, Yusuke Kobayashi, Joshua J. Kennedy-Smith,
F. Dean Toste* Chemistry – A European Journal, 16 (31), 9555–9562 (2010) |
HTLV-1 basic leucine-zipper
factor, HBZ, interacts with MafB and suppresses transcription through a Maf
recognition element Takayuki
Ohshima,* Risa Mukai, Norie Nakahara, Jun Matsumoto, Osamu Isono, Yusuke
Kobayashi, Satoru Takahashi, Kunitada Shimotohno Journal of Cellular Biochemistry, 111 (1), 187–194
(2010) |
Effects of sulfaphenazole derivatives
on cardiac ischemia–reperfusion injury: association of cytochrome P450 activity
and infarct size Yasuhiro
Ishihara, Masaya Sekine, Ai Hamaguchi, Yusuke Kobayashi, Takashi
Harayama, Mikio Nakazawa, Norio Shimamoto* Journal of Pharmacological
Sciences,
113, 335 – 342 (2010) |
Trifluoroacetylation-induced
Houben−Hoesch-type cyclization of cyanoacetanilides: increased nucleophilicity
of CN groups Yusuke
Kobayashi,*
Kosuke Katagiri, Isao Azumaya and Takashi Harayama The Journal of Organic Chemistry, 75 (8), 2741–2744 (2010) |